Recently, xanthones are found to be interesting due to their diverse pharmacological activities. Although xanthones can obtained and isolated from natural products and through biosynthesis of natural products, but the studies of synthesized xanthones by laboratory skills are more focused since years back. The main reason why there is an increase interest in chemical synthesis is that synthetic approach can afford to prepare different type of xanthones with diverse structure. Moreover, through chemical synthesis, the percent yield of synthesized xanthones can be increased.